Protein detail

IDE

Insulin-degrading enzyme (EC 3.4.24.56) (Abeta-degrading protease) (Insulin protease) (Insulinase) (Insulysin)

Protein symbol
IDE
UniProt ID
EVMP score
0.38
Frequency
Transmembrane count
Protein classification
EnzymesFDA approved drug targetsPlasma proteinsPredicted intracellular proteinsPredicted secreted proteins
Basic Information
Protein Names
Insulin-degrading enzyme (EC 3.4.24.56) (Abeta-degrading protease) (Insulin protease) (Insulinase) (Insulysin)
Protein Class
EnzymesFDA approved drug targetsPlasma proteinsPredicted intracellular proteinsPredicted secreted proteins
Protein Function
  • Predicted intracellular proteins
  • Enzymes
  • Predicted secreted proteins
  • ENZYME proteins:Hydrolases
  • Peptidases:Metallopeptidases
  • FDA approved drug targets:Small molecule drugs
Entrez Gene Symbol
Gene Description
Insulin degrading enzyme
Chromosome
10
Position
92451684-92574096
EVMP Score
0.38
Fluorescence & Localization
Cell SpecificBrain excitatory neuronsSingle-Nuclei Brain Specificlower rhombic lipBlood Cell SpecificMAIT T-cellBlood Lineage SpecificT-cells
Function & Pathway
Protein Function
  • Predicted intracellular proteins
  • Enzymes
  • Predicted secreted proteins
  • ENZYME proteins:Hydrolases
  • Peptidases:Metallopeptidases
  • FDA approved drug targets:Small molecule drugs
Mediation Categories
Clinical-translation mediationFusion and delivery mediationImmune mediationMetabolism mediationReceptor-signaling mediation
Relations & Evidence

Enzyme-Mediated Modification

0 records.

Ligand-Receptor Signaling

22 records.

CategoryParentDatabaseTransmitterReceiverSecretedPlasma Membrane (Transmembrane)Plasma Membrane (Peripheral)
intracellularintracellularOmniPathNoNoYesNoNo
insulin_degradingcell_surface_peptidaseOmniPathYesNoYesNoNo
m16_metallopeptidasecell_surface_peptidaseOmniPathYesNoYesNoNo
cell_surface_enzymecell_surface_enzymeOmniPathYesNoYesNoNo
cell_surface_peptidasecell_surface_peptidaseOmniPathYesNoYesNoNo
secreted_peptidasesecreted_peptidaseOmniPathNoNoYesNoNo
plasma_membraneplasma_membraneUniProt_locationNoNoYesNoNo
plasma_membraneplasma_membraneOmniPathNoNoYesNoNo
secretedsecretedUniProt_keywordNoNoYesNoNo
secretedsecretedUniProt_locationNoNoYesNoNo
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Regulatory Interaction Network

1 record.

Source Protein SymbolSource UniProt IDTarget Protein SymbolTarget UniProt IDIs DirectedIs StimulationIs InhibitionDatabaseReferences
IDEP14735INSP01308YesNoYesSIGNORHPRDHINTIntActDIPHINT:19321446HINT:29273204HPRD:11145591HPRD:17051221HINT:17051221IntAct:17051221HINT:29596046SIGNOR:29596046DIP:17051221

Protein Complex Composition

26 records.

Component NameComponent Gene SymbolsComponent UniProt IDStoichiometryDatabaseDatabase IDsReferences
HT_DM_Cluster473CIDEACIDEBCIDECSRMO60543P19623Q96AQ7Q9UHD41:1:1:1CompleatCompleat:HC351322036573
HT_SC_Cluster373IDENRDCSPENO43847P14735Q96T581:1:1CompleatCompleat:HC1808
MiDAC complexDNTTIP1HDAC1HDAC2MIDEASQ13547Q6PJG2Q92769Q9H1470:0:0:0CORUMCORUM:637321258344
MiDAC histone deacetylase complexHDAC1 variantDNTTIP1HDAC1MIDEASQ13547Q6PJG2Q9H1472:2:2ComplexPortalPDBPDB:6z2jPDB:6z2kintact:EBI-9027309147552922565316532591534
MiDAC histone deacetylase complexHDAC2 variantDNTTIP1HDAC2MIDEASQ6PJG2Q92769Q9H1471:1:1ComplexPortalintact:EBI-9027193147552922565316532591534
CHD1LDNM2H2AXH2BC12H3-3AH4C4HMGB1HMGB2IDEPRKDCRPA1SMARCA4SMARCA5O60264O60814P09429P14735P16104P26583P27694P50570P51532P62805P78527P84243Q86WJ11:1:1:1:1:1:1:1:1:1:1:1:1NetworkBlastCompleatCompleat:HC9390
IDETGFAP01135P147352:2PDBPDB:3e50
IDENPPAP01160P147352:2PDBPDB:3n57
GCGIDEP01275P147352:2PDBPDB:2g49PDB:6eds
IDEINSP0DOX5Q6GMX0P01308P0DOX5P14735Q6GMX02:2:2:2PDBPDB:6b70
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Isolation & Detection Technology

1 record.

EV Isolation MethodDetection MethodNumber of ReferencesReferences
Differential UltracentrifugationSize Exclusion ChromatographyMass spectrometry132331267
Sequence, Structure & Domains

Sequences

Length
1,019
Mass
117,968
Sequence
MRYRLAWLLHPALPSTFRSVLGARLPPPERLCGFQKKTYSKMNNPAIKRIGNHITKSPEDKREYRGLELANGIKVLLISDPTTDKSSAALDVHIGSLSDPPNIAGLSHFCEHMLFLGTKKYPKENEYSQFLSEHAGSSNAFTSGEHTNYYFDVSHEHLEGALDRFAQFFLCPLFDESCKDREVNAVDSEHEKNVMNDAWRLFQLEKATGNPKHPFSKFGTGNKYTLETRPNQEGIDVRQELLKFHSAYYSSNLMAVCVLGRESLDDLTNLVVKLFSEVENKNVPLPEFPEHPFQEEHLKQLYKIVPIKDIRNLYVTFPIPDLQKYYKSNPGHYLGHLIGHEGPGSLLSELKSKGWVNTLVGGQKEGARGFMFFIINVDLTEEGLLHVEDIILHMFQYIQKLRAEGPQEWVFQECKDLNAVAFRFKDKERPRGYTSKIAGILHYYPLEEVLTAEYLLEEFRPDLIEMVLDKLRPENVRVAIVSKSFEGKTDRTEEWYGTQYKQEAIPDEVIKKWQNADLNGKFKLPTKNEFIPTNFEILPLEKEATPYPALIKDTAMSKLWFKQDDKFFLPKACLNFEFFSPFAYVDPLHCNMAYLYLELLKDSLNEYAYAAELAGLSYDLQNTIYGMYLSVKGYNDKQPILLKKIIEKMATFEIDEKRFEIIKEAYMRSLNNFRAEQPHQHAMYYLRLLMTEVAWTKDELKEALDDVTLPRLKAFIPQLLSRLHIEALLHGNITKQAALGIMQMVEDTLIEHAHTKPLLPSQLVRYREVQLPDRGWFVYQQRNEVHNNCGIEIYYQTDMQSTSENMFLELFCQIISEPCFNTLRTKEQLGYIVFSGPRRANGIQGLRFIIQSEKPPHYLESRVEAFLITMEKSIEDMTEEAFQKHIQALAIRRLDKPKKLSAECAKYWGEIISQQYNFDRDNTEVAYLKTLTKEDIIKFYKEMLAVDAPRRHKVSVHVLAREMDSCPVVGEFPCQNDINLSQAPALPQPEVIQNMTEFKRGLPLFPLVKPHINFMAAKL
Alternative Products
Event=Alternative splicing; Named isoforms=2; Name=1; IsoId=P14735-1; Sequence=Displayed; Name=2; IsoId=P14735-2; Sequence=VSP_044303
Alternative Sequence
1..555; Missing (in isoform 2)

3D Structural Models

Turn
133..135; 326..328; 441..443; 449..454; 486..488; 494..496; 824..827
Helix
96..98; 106..113; 114..116; 126..132; 155..157; 158..166; 167..169; 176..194; 197..207; 214..216; 223..226; 228..232; 237..248; 251..253; 264..275; 295..297; 323..325; 330..338; 346..352; 381..385; 387..404; 408..423; 430..440; 446..448; 461..468; 473..475; 483..485; 507..514; 581..583; 587..613; 638..650; 656..672; 673..675; 678..690; 697..704; 709..721; 735..753; 760..762; 802..823; 856..876; 879..894; 900..912; 920..928; 933..943; 995..1000
Beta Strand
47..50; 63..69; 74..79; 84..93; 101..104; 118..121; 123..125; 137..142; 147..154; 254..262; 276..278; 298..304; 307..309; 312..319; 359..367; 370..378; 477..481; 499..504; 549..553; 555..563; 565..567; 570..579; 584..586; 616..623; 626..635; 691..693; 722..732; 775..782; 787..799; 831..840; 843..854; 945..947; 949..951; 952..959; 990..992
3D Structure
Electron microscopy (14); X-ray crystallography (47)

Domain & Motif Annotations

Motif
853..858; SlyX motif
Domain (CC)
The SlyX motif may be involved in the non-conventional secretion of the protein.
Protein Families
Peptidase M16 family
Sequence Similarities
Belongs to the peptidase M16 family.
Clinical Relevance
Disease Involvement
FDA approved drug targets
Biomarker
Phase 2; Approved
Drug Targets
FDA approved drug targets
Antibody
Interaction Protein
ENSG00000089163
Interaction Count
1
Interaction Dataset
intact_biogrid