Protein detail

TACD2

Tumor-associated calcium signal transducer 2 (Cell surface glycoprotein Trop-2) (Membrane component chromosome 1 surface marker 1) (Pancreatic carcinoma marker protein GA733-1)

Entry name
TACD2
UniProt ID
EVMP confidence score
0.72
Supporting publications (n)
16
Transmembrane count
1
Protein classification
Disease related genesFDA approved drug targetsHuman disease related genesPredicted membrane proteins
EVMP confidence score

Annotation confidence score; open for threshold definitions.

Extremely high >= 0.85High >= 0.70Medium >= 0.55Low >= 0.40
Basic Information13
Protein Names
Tumor-associated calcium signal transducer 2 (Cell surface glycoprotein Trop-2) (Membrane component chromosome 1 surface marker 1) (Pancreatic carcinoma marker protein GA733-1)
Protein Class (4)
Disease related genesFDA approved drug targetsHuman disease related genesPredicted membrane proteins
Protein Function (3)
  • Disease related genes
  • Human disease related genes:Nervous system diseases:Eye disease
  • FDA approved drug targets:Biotech drugs
Transmembrane
275..297; Helical
Transmembrane Count
1
Entrez Gene Symbol
Gene Synonym (4)
EGP-1GA733-1M1S1TROP2
Gene Description
Tumor associated calcium signal transducer 2
Chromosome
1
Position
58575433-58577252
Supporting publications (n)
16
EVMP confidence score
0.72
Function & Pathway5
Protein Function (3)
  • Disease related genes
  • Human disease related genes:Nervous system diseases:Eye disease
  • FDA approved drug targets:Biotech drugs
Mediation Categories (3)
Adhesion and uptake mediationClinical-translation mediationFusion and delivery mediation
Relations & Evidence31

Enzyme-Mediated Modification (3)

3 records.

Substrate Gene SymbolEnzyme Gene SymbolEnzyme UniProt IDResidue TypeResidue OffsetModificationDatabaseReferences
TACSTD2PRKCAP17252S303phosphorylationPhosphoNetworksphosphoELM_MIMPPhosphoSite_MIMPMIMPProtMapperKEAphosphoELMPhosphoSitePhosphoSite_ProtMapperphosphoELM:7635574KEA:7635574
TACSTD2PRKCAP17252S322phosphorylationPhosphoSite
TACSTD2PRKCDQ05655S322phosphorylationPhosphoSite

Ligand-Receptor Signaling (23)

23 records.

CategoryParentDatabaseTransmitterReceiverSecretedPlasma Membrane (Transmembrane)Plasma Membrane (Peripheral)
transmembranetransmembraneRamilowski_locationNoNoNoYesNo
transmembranetransmembraneOmniPathNoNoNoYesNo
plasma_membrane_transmembraneplasma_membrane_transmembraneMembranomeNoNoNoYesNo
plasma_membrane_transmembraneplasma_membrane_transmembraneCSPANoNoNoYesNo
plasma_membrane_transmembraneplasma_membrane_transmembraneOmniPathNoNoNoYesNo
cell_surfacecell_surfaceSurfaceomeNoNoNoYesNo
cell_surfacecell_surfaceOmniPathNoNoNoYesNo
receptorreceptorscConnectNoYesNoYesNo
receptorreceptorCellCellInteractionsNoYesNoYesNo
transmembranetransmembrane_predictedPhobiusNoNoNoYesNo
Page 2 of 3PreviousNext

Regulatory Interaction Network (3)

3 records.

Source Protein SymbolSource UniProt IDTarget Protein SymbolTarget UniProt IDIs DirectedIs StimulationIs InhibitionDatabaseReferences
KPCDQ05655TACD2P09758YesNoYesSIGNORPhosphoSite_ProtMapperProtMapperSIGNOR:31177095
TACD2P09758CLD7O95471YesYesNoHINTLit-BM-17SIGNORLit-BM-17:20651236HINT:20651236SIGNOR:31177095HINT:33961781
KPCAP17252TACD2P09758YesNoYesPhosphoNetworksphosphoELM_MIMPPhosphoSite_MIMPMIMPiPTMnetSIGNORProtMapperPhosphoSite_KEAKEAphosphoELM_KEAphosphoELMPhosphoSitePhosphoSite_ProtMapperKEA:7635574phosphoELM:7635574SIGNOR:31177095PhosphoSite:31177095PhosphoSite:25981199PhosphoSite:7635574

Protein Complex Composition (1)

1 record.

Component NameComponent Gene SymbolsComponent UniProt IDStoichiometryDatabaseDatabase IDsReferences
TACSTD2P097582PDBPDB:7e5nPDB:7e5mPDB:7pee

Isolation & Detection Technology (1)

1 record.

EV Isolation MethodDetection MethodNumber of ReferencesReferences
Differential UltracentrifugationSize Exclusion ChromatographyMass spectrometry130865381
Sequence, Structure & Domains10

Sequences

Length
323
Mass
35,709
Sequence
MARGPGLAPPPLRLPLLLLVLAAVTGHTAAQDNCTCPTNKMTVCSPDGPGGRCQCRALGSGMAVDCSTLTSKCLLLKARMSAPKNARTLVRPSEHALVDNDGLYDPDCDPEGRFKARQCNQTSVCWCVNSVGVRRTDKGDLSLRCDELVRTHHILIDLRHRPTAGAFNHSDLDAELRRLFRERYRLHPKFVAAVHYEQPTIQIELRQNTSQKAAGDVDIGDAAYYFERDIKGESLFQGRGGLDLRVRGEPLQVERTLIYYLDEIPPKFSMKRLTAGLIAVIVVVVVALVAGMAVLVITNRRKSGKYKKVEIKELGELRKEPSL

3D Structural Models

Turn
58..60; 121..123
Helix
49..51; 72..80; 169..182; 188..190; 209..211; 219..230; 299..317
Beta Strand
41..46; 54..57; 97..99; 112..114; 116..120; 124..129; 151..160; 191..197; 200..206; 237..239; 253..264
3D Structure
NMR spectroscopy (3); X-ray crystallography (3)

Domain & Motif Annotations

Domain (FT)
70..145; Thyroglobulin type-1
Protein Families
EPCAM family
Sequence Similarities
Belongs to the EPCAM family.
Clinical Relevance6
Disease Involvement (3)
AmyloidosisCorneal dystrophyFDA approved drug targets
Biomarker
Approved; Phase 3; Phase 1/2
Drug Targets
FDA approved drug targets
Supporting Publications16
PMIDTitleAbstract
23161513Proteomic analysis of exosomes from mutant KRAS colon cancer cells identifies intercellular transfer of mutant KRAS.Exosomes from mutant KRAS cells contain many tumor-promoting proteins, including KRAS, EGFR, SRC family kinases, and integrins.
27894104Proteomic profiling of NCI-60 extracellular vesicles uncovers common protein cargo and cancer type-specific biomarkers.No abstract available
28986585Quantitation of putative colorectal cancer biomarker candidates in serum extracellular vesicles by targeted proteomics.No abstract available
29045505Surfaceome profiling enables isolation of cancer-specific exosomal cargo in liquid biopsies from pancreatic cancer patients.Proteomic analysis of the exosome 'surfaceome' revealed multiple PDAC-specific biomarker candidates: CLDN4, EPCAM, CD151, LGALS3BP, HIST2H2BE, and HIST2H2BF. Droplet digital PCR was used on 74 patients (136 total exosome samples) to determine baseline KRAS mutation call rates while patients were on therapy. KRAS mutations in total exosomes were detected in 44.1% of patients undergoing active therapy compared with 73.0% following exosome capture using the selected biomarkers.
30379855Harmonization of exosome isolation from culture supernatants for optimized proteomics analysis.No abstract available
30646616Preferential Localization of MUC1 Glycoprotein in Exosomes Secreted by Non-Small Cell Lung Carcinoma Cells.THBS1, ANXA6, HIST1H4A, COL18A1, MDK, SRGN, ENO1, TUBA4A, SLC3A2, GPI, MIF, MUC1, TALDO1, SLC7A5, ICAM1, HSP90AA1, G6PD, and LRP1 were found to be expressed in exosomes at more than 5-fold higher level as compared to total cellular membrane proteins.
30950185Unique Protein Profiles of Extracellular Vesicles as Diagnostic Biomarkers for Early and Advanced Non-Small Cell Lung Cancer.No abstract available
32284825Unravelling the proteomic landscape of extracellular vesicles in prostate cancer by density-based fractionation of urine.No abstract available
34186243A Reductionist Approach Using Primary and Metastatic Cell-Derived Extracellular Vesicles Reveals Hub Proteins Associated with Oral Cancer Prognosis.No abstract available
34571828Proteomic Analysis of Circulating Extracellular Vesicles Identifies Potential Biomarkers for Lymph Node Metastasis in Oral Tongue Squamous Cell Carcinoma.No abstract available
Page 1 of 2Next