Protein detail

S22A8

Organic anion transporter 3 (hOAT3) (Organic anion/dicarboxylate exchanger) (Solute carrier family 22 member 8)

Protein symbol
S22A8
UniProt ID
EVMP score
0.38
Frequency
Transmembrane count
11
Protein classification
FDA approved drug targetsMetabolic proteinsPredicted membrane proteinsTransporters
Basic Information
Protein Names
Organic anion transporter 3 (hOAT3) (Organic anion/dicarboxylate exchanger) (Solute carrier family 22 member 8)
Protein Class
FDA approved drug targetsMetabolic proteinsPredicted membrane proteinsTransporters
Protein Function
  • Transporters:Electrochemical Potential-driven transporters
  • FDA approved drug targets:Small molecule drugs
Transmembrane
10..30; Helical; 124..144; Helical; 155..175; Helical; 177..197; Helical; 213..233; Helical; 237..257; Helical; 328..348; Helical; 355..375; Helical; 387..407; Helical; 412..432; Helical; 472..492; Helical
Transmembrane Count
11
Entrez Gene Symbol
Gene Synonym
OAT3
Gene Description
Solute carrier family 22 member 8
Chromosome
11
Position
62989154-63015841
EVMP Score
0.38
Fluorescence & Localization
Cell SpecificFibro-adipogenic progenitorsSingle-Nuclei Brain Specificoligodendrocyte
Function & Pathway
Relations & Evidence

Enzyme-Mediated Modification

0 records.

Ligand-Receptor Signaling

20 records.

CategoryParentDatabaseTransmitterReceiverSecretedPlasma Membrane (Transmembrane)Plasma Membrane (Peripheral)
receptorreceptorOmniPathNoYesNoNoNo
transportertransporterSurfaceomeNoYesNoNoNo
mfstransporterSurfaceomeNoYesNoNoNo
slc22transporterSurfaceomeNoYesNoNoNo
slctransporterSurfaceomeNoYesNoNoNo
transportertransporterOmniPathNoYesNoNoNo
transmembranetransmembraneUniProt_locationNoNoNoNoNo
transmembranetransmembraneUniProt_topologyNoNoNoNoNo
transmembranetransmembraneUniProt_keywordNoNoNoNoNo
transmembranetransmembraneRamilowski_locationNoNoNoNoNo
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Regulatory Interaction Network

0 records.

Protein Complex Composition

0 records.

Isolation & Detection Technology

1 record.

EV Isolation MethodDetection MethodNumber of ReferencesReferences
Differential UltracentrifugationUltrafiltration / Tangential Flow FiltrationSize Exclusion ChromatographyImmunoaffinity CaptureMass spectrometry143371834237862381389386743994949026538482315085003887173037702715327954143007131837033249376863664009834633114768
Sequence, Structure & Domains

Sequences

Length
542
Mass
59,856
Sequence
MTFSEILDRVGSMGHFQFLHVAILGLPILNMANHNLLQIFTAATPVHHCRPPHNASTGPWVLPMGPNGKPERCLRFVHPPNASLPNDTQRAMEPCLDGWVYNSTKDSIVTEWDLVCNSNKLKEMAQSIFMAGILIGGLVLGDLSDRFGRRPILTCSYLLLAASGSGAAFSPTFPIYMVFRFLCGFGISGITLSTVILNVEWVPTRMRAIMSTALGYCYTFGQFILPGLAYAIPQWRWLQLTVSIPFFVFFLSSWWTPESIRWLVLSGKSSKALKILRRVAVFNGKKEEGERLSLEELKLNLQKEISLAKAKYTASDLFRIPMLRRMTFCLSLAWFATGFAYYSLAMGVEEFGVNLYILQIIFGGVDVPAKFITILSLSYLGRHTTQAAALLLAGGAILALTFVPLDLQTVRTVLAVFGKGCLSSSFSCLFLYTSELYPTVIRQTGMGVSNLWTRVGSMVSPLVKITGEVQPFIPNIIYGITALLGGSAALFLPETLNQPLPETIEDLENWSLRAKKPKQEPEVEKASQRIPLQPHGPGLGSS
Alternative Products
Event=Alternative splicing; Named isoforms=5; Name=1; IsoId=Q8TCC7-1; Sequence=Displayed; Name=2; IsoId=Q8TCC7-2; Sequence=VSP_022565; Name=5; IsoId=Q8TCC7-5; Sequence=VSP_045824; Name=3; IsoId=Q8TCC7-3; Sequence=VSP_022562, VSP_022563, VSP_022564; Name=4; IsoId=Q8TCC7-4; Sequence=VSP_045272
Alternative Sequence
1..345; Missing (in isoform 3); 1..123; Missing (in isoform 5); 1..91; Missing (in isoform 4); 406..455; DLQTVRTVLAVFGKGCLSSSFSCLFLYTSELYPTVIRQTGMGVSNLWTRV -> GERLGLPQNPLEEAARLGARDFTAGSASKSLCYLEQVPALSGAQGLSSRK (in isoform 3); 456..542; Missing (in isoform 3); 510; W -> WSVTASGPPR (in isoform 2)

3D Structural Models

Domain & Motif Annotations

Compositional Bias
517..527; Basic and acidic residues
Region
515..542; Disordered
Protein Families
  • Major facilitator (TC 2.A.1) superfamily
  • Organic cation transporter (TC 2.A.1.19) family
Sequence Similarities
Belongs to the major facilitator (TC 2.A.1) superfamily. Organic cation transporter (TC 2.A.1.19) family.
Clinical Relevance